英语词根词缀记忆大全 (2).doc
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1、倘(琀币匀爀币币琀币讀缁缀劙漁螏頀h椀霂褃匃匈匈漈茈謈謈謈嘀一一刀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀瀀椀挀最椀昀嘀一一刀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀尀尀戀昀搀昀挀挀攀攀昀愀攀戀愀挀儀猀一栀砀愀最椀堀儀嘀瀀唀搀眀氀挀堀匀伀猀洀堀嘀唀倀琀昀栀堀眀刀欀爀甀稀樀瘀眀嘀一一刀攀搀栀攀洀砀瀀爀攀猀猀愀挀昀愀昀挀攀挀搀瀀瀀洀琀愀琀攀甀最漀挀甀洀攀渀琀猀吀椀琀氀攀愀琀愀氀漀最一漀夀愀琀挀栀匀瀀攀挀琀爀甀洀吀椀琀氀攀夀开娀圀夀儀爀攀焀甀攀渀挀礀稀昀伀爀椀最椀渀愀氀倀漀椀渀琀猀漀甀渀琀昀挀琀甀愀氀倀漀椀渀琀猀漀甀渀琀昀挀焀甀椀猀椀琀椀漀渀吀椀洀攀猀攀挀昀匀瀀攀挀琀爀愀氀圀椀搀琀栀瀀瀀洀昀倀甀氀猀攀倀爀漀最爀愀洀唀渀欀渀
2、漀眀渀匀愀洀瀀氀攀娀圀夀儀愀琀愀氀漀最一漀夀愀琀挀栀匀伀匀伀伀一一一一一栀攀洀椀挀愀氀漀爀洀甀氀愀一伀匀砀愀挀琀愀猀猀攀搀栀攀洀砀瀀爀攀猀猀靓辉退舀祒茤佦蠀懈!牁鄃凍艉芓蕞庂膅!牁鄃凍蝉芓蕞庂膅!牁鄃勍艑芓皫腶!牁鄃勍蝑芓皫腶!鄊勍芛芓琀挛匜褛鬛猞鄚1芪!騀苻1鳚芬!攀倐猠舐魒鎇者跥t鴡蠡裭頀苙!頀苻!芜!鏟!e瀐酐魒嵗鎂苤魒嵗鎇苤灓鎂苅灓鎇苅鄀鎂艡仉偐İ!跮鰀!鄅反蟠芓懒荎!馜鎂肅藎牁鄄囍蟴肓藎膅!脀譗鎂脶鬏+苯鬡頞鰘譗鎇脶鬏+苯鬡頞鰘腐鎂嚂胴,騱臈!脀舐脐鄊姍蜍芓褍踡灰怐鄊姍舧芓贄褙蠡抺輛雾鈡拝抚鏝蓈輐铿鼡鸟努鬡!倄鉐脐怐灠瀠【灀鄰怐偰灀偀Q|鄊姍蜧芓贄褙蠡抺輛雾鈡拝抚鏝蓈輐铿鼡鸟努鬡!倄
3、艐偀怐【Lw鄅巍若芓庁茨辍闞鎇脰辍!牁鄄巍以舚肓膾1脀鎇肾虞鎂鈃臖贜頡勍叹臹爛颙鯩釸拏輚萡訡力勎鐡贱香謟蒫舟蠐蓛踡拏鸐霝蔱鄘鬜覜頡勹裘鬐鄡袚鋏頡拪鼏势挚h倁倠恠恠恠恠恠扠恠恠恠扠倰偐偀瀐瀁倠倐唀紀省鼁朂鄂尃虞鎇鈃臖贜頡勍勹醹臸餉鏊馮輡鯹鼏蘡鰡力勎鐡贡香膽蒫钺犎谛谐钿拏霝蔡鄘鬜覜頡闿兄(币搀爀币币币讀缁缀劜漁螏頀h椀圃圃圃霃匀愀琀愀匀栀攀攀琀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀瀀椀挀最椀昀匀愀琀愀匀栀攀攀琀攀搀栀攀洀砀瀀爀攀猀猀瀀搀昀尀尀愀戀戀挀搀搀戀戀攀戀攀昀挀愀昀伀洀搀攀氀匀搀嘀圀爀刀戀椀爀欀唀渀漀戀椀爀砀唀儀最最椀刀瘀最眀匀愀琀愀匀栀攀攀琀攀搀栀攀洀砀瀀爀攀猀猀昀戀愀昀攀昀昀挀搀Z屇攀搀栀攀洀砀瀀
4、爀攀猀猀靓 schedule (100-300 mpk) or a twice a day schedule (50, 100 mpk) demonstrates antitumor activity in this tumor model. Oral glucose tolerance test (OGTT) shows 100 mpk (b.i.d.) causes a significant DescriptionProduct Data Sheet InhibitorsAgonistsScreening Librarieswww.MedChemE1elevation in glucos
5、e levels after glucose challenge. The pharmacokinetic parameters of BMS-536924, administered orally in poly(ethylene glycol) 400 and water (80:20 v/v), are determined in mouse, rat, dog, and monkey. Good bioavailability is evident in all species. Significant nonlinear pharmacokinetics is observed in
6、 rodents at increasing p.o. dose 1. Oral administration of 70 mg/kg BMS-536924 significantly inhibits tumor growth (TGBC-1TKB cells) inoculated in nude mice. BMS-536924 up regulates apoptosis in xenografts tumors. The treatment doesnt have adverse effects on the body weight of mice or the glucose le
7、vels at the time of death, suggesting tolerable toxicity 3.REFERENCES1. Wittman M, et al. Discovery of a (1H-benzoimidazol-2-yl)-1H-pyridin-2-one (BMS-536924) inhibitor of insulin-like growth factor I receptor kinase with in vivo antitumor activity. J Med Chem. 2005 Sep 8;48(18):5639-43.2. Litzenbur
8、ger BC, et al. BMS-536924 reverses IGF-IR-induced transformation of mammary epithelial cells and causes growth inhibition and polarization of MCF7 cells. Clin Cancer Res. 2009 Jan 1;15(1):226-37.3. Ohashi H, et al. Insulin-like growth factor receptor expression is associated with aggressive phenotyp
9、es and has therapeutic activity in biliary tract cancers. Cancer Sci. 2012 Feb;103(2):252-61.Caution: Product has not been fully validated for medical applications. For research use only.Tel: 609-228-6898 Fax: 609-228-5909 E-mail: techMedChemEAddress: 1 Deer Park Dr, Suite Q, Monmouth Junction, NJ 0
10、8852, USAwww.MedChemE2MedChemExpress0001500006先进医疗20190531141510815982辉退舀祒茤佦蠀懈!牁鄃凍艉芓蕞庂膅!牁鄃凍蝉芓蕞庂膅!牁鄃勍艑芓皫腶!牁鄃勍蝑芓皫腶!鄊勍芛芓琀挛匜褛鬛猞鄚1芪!騀苻1鳚芬!攀倐猠舐魒鎇者跥t鴡蠡裭頀苙!頀苻!芜!鏟!e瀐酐魒嵗鎂苤魒嵗鎇苤灓鎂苅灓鎇苅鄀鎂艡仉偐İ!跮鰀!鄅反蟠芓懒荎!馜鎂肅藎牁鄄囍蟴肓藎膅!脀譗鎂脶鬏+苯鬡頞鰘譗鎇脶鬏+苯鬡頞鰘腐鎂嚂胴,騱臈!脀舐脐鄊姍蜍芓褍踡灰怐鄊姍舧芓贄褙蠡抺輛雾鈡拝抚鏝蓈輐铿鼡鸟努鬡!倄鉐脐怐灠瀠【灀鄰怐偰灀偀Q|鄊姍蜧芓贄褙蠡抺輛雾鈡拝抚鏝蓈輐铿鼡鸟努鬡!倄艐
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