A-839977-DataSheet-MedChemExpress.pdf
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1、A 839977Cat. No.: HY-13954CAS No.: 870061-27-1Molecular Formula: CHClNOMolecular Weight: 413.26Target: P2X ReceptorPathway: Membrane Transporter/Ion ChannelStorage: Powder -20C 3 years4C 2 yearsIn solvent -80C 6 months-20C 1 monthSolvent blocks BzATP-evoked calcium influx at recombinant human, rat a
2、nd mouse P2X7 receptors (IC50 values are 20, 42 and 150 nM respectively).IC50 Value: Target: P2X7in vitro: A-839977 potently (IC50=20-150 nM) blocked BzATP-evoked calcium influx at recombinant human, rat and mouse P2X7 receptors. A-839977 also potently blocked agonist-evoked YO-PRO uptake and IL-1be
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- 839977 DataSheet MedChemExpress